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- Volynets
GP, Chekanov OM, Synyugin AR, Golub AG, Kukharenko OP, Bdzhola VG,
Yarmoluk SM. Identification of 3H-naphtho[1,2,3-de]quinoline-2,7-diones
as inhibitors of apoptosis signal-regulating kinase 1 (ASK1) http://pubs.acs.org/doi/abs/10.1021/jm200117h
-
Golub AG, Bdzhola VG, Briukhovetska NV, Balanda AO, Kukharenko OP,
Kotey IM, Ostrynska OV, Yarmoluk SM. Synthesis and biological evaluation
of substituted (thieno[2,3-d]pyrimidin-4-ylthio)carboxylic acids as
inhibitors of human protein kinase CK2. Eur. J. Med. Chem. 2011 Mar;
46(3): 870-6.
- Volynets GP,
Bdzhola VG, Kukharenko OP, Yarmoluk SM. Identification of ASK1 small-molecule
inhibitors. Ukr. Biochim. J. 2010; 82 (5): 26-34.
- Grischenko AA,
Bdzhola VG, Kukharenko OP, Yarmoluk SM. Search for FGFR1 inhibitors
among chromone derivatives. Ukrainica Bioorganica Acta. 2009; 7 (2):
64-68.
- Kotey IM, Balanda
AO, Bdzhola VG, Lukashov SS, Kukharenko OP, Kharchenko VM, Yarmoluk
SM. Synthesis and biologic evaluation of thienopyrimidinones inhibition
activity against protein kinase CK2. Ukrainica Bioorganica Acta. 2008.
6 (2): 3-9.
- Grischenko AA,
Bdzhola VG, Kukharenko OP, Yarmoluk SM. Search for FGFR1 inhibitors
among chromone derivatives. Ukrainica Bioorganica Acta. 2009. 7 (1):
50-56.
- Volynets GP,
Bdzhola VG, Yarmoluk SM. Methods of structural bioinformatics. Biotechnology.
2010; 3 (4): 9-19.
- Volynets GP,
Bdzhola VG, Kukharenko OP, Sovetova OV, Yarmoluk SM. Protein kinase
ASK1 as potential therapeutic target. Biopolymers and Cell. 2009.
25 (3): 169-180.
- Project: STSU-NASU
¹ 5218 Rational search for inhibitors of aminoacyl-tRNA synthetases
with selective action against causative agent of tuberculosis 2010-2012.
- Volkova
KD, Kovalska VB, Balanda AO, Losytskyy MY, Golub AG, Vermeij RJ, Subramaniam
V, Tolmachev OI, Yarmoluk SM. Specific fluorescent detection of fibrillar
alpha-synuclein using mono- and trimethine cyanine dyes. Bioorg Med
Chem. 2008 Feb 1;16(3):1452-9.
- Golub AG, Yakovenko
OY, Prykhod'ko AO, Lukashov SS, Bdzhola VG, Yarmoluk SM. Evaluation
of 4,5,6,7-tetrahalogeno-1H-isoindole-1,3(2H)-diones as inhibitors
of human protein kinase CK2. Biochim Biophys Acta. 2008 Jan;1784(1):143-9.
- Yakovenko O,
Oliferenko AA, Bdzhola VG, Palyulin VA, Zefirov NS. Kirchhoff atomic
charges fitted to multipole moments: implementation for a virtual
screening system. J Comput Chem. 2008 Jun;29(8):1332-43.
- Golub AG, Yakovenko
OY, Bdzhola VG, Sapelkin VM, Zien P, Yarmoluk SM. Evaluation of 3-carboxy-4(1H)-quinolones
as inhibitors of human protein kinase CK2. J Med Chem. 2006 Nov 2;49(22):6443-50.
- Yakovenko. O.Ya.,
Oliferenko A.A., Golub G.A., Bdzhola V.G., Yarmoluk S.M. The new method
of distribution integrals evaluations for high throughput virtual
screening. / Ukrainica Bioorganica Acta, Vol5 N1 2007, P52-63.
- Yakovenko. O.Ya.,
Golub G.A., Bdzhola V.G., Yarmoluk S.M. Application of distribution
function of rotation and translation degrees of freedom for CK2 inhibitors
Ki estimation. / Ukrainica Bioorganica Acta, Vol4 N2 2006, P47-56.
- Sapelkin V.,Yakovenko
O.,Golub A., Bdzhola V., Yarmoluk S. Search for protein kinase CK2
inhibitors among 3 carbetoxy 4 aminoquinoline derivatives. Ukrainica
Bioorganica Acta. 2005. – 2, ¹ 1, 28-32.
- Prykhod'ko A.O.,
Yakovenko O.Ya., Golub A.G., Bdzhola V. G., Yarmoluk S.M. Evaluation
of 4H-4-chromenone derivatives as inhibitors of protein kinase CK2.
Biopolymers and Cell, 2005. – 21, ¹ 3, 287-292.
- Golub A.G., Yakovenko
O.Ya., Bdzhola V. G., Yarmoluk S.M. Implementation of orbital graph
model for partial atom charges definition in virtual screening techniques.
Cell. Mol. Biol. Lett. – Vol. 10, N 2A. – 2005. – P. 126.
- Golub A.G.,
Yakovenko O.Ya., Sapelkin V.M., Bdzhola V. G., Yarmoluk S.M. Evaluation
of 3-carboxy-4-(1H)-quinolones as inhibitors of human protein casein
kinase 2. Cell. Mol. Biol. Lett. – Vol. 10, N 2A. – 2005. – P. 102.
- Pat. UÀ68984
À, C07D215/00, 2004-08-16. Application of 4-substituted 3-carboxyquinolines
as protein kinase CK2 inhibitors. Sapelkin V.M., Lukashov S.S., Golub
A.G., Bdzhola V. G., Yakovenko O.Ya., Yarmoluk S.M., Dubinina G.G.
- Pat. UA69165
À, Ñ07D215/00, 2004-08-16. Application of 4,5,6,7-tetrahalogeno-1,3-isoindolinediones
as protein kinase CK2 inhibitors. Golub A.G., Yakovenko O.Ya., Yarmoluk
S.M., Dubinina G.G., Bdzhola V. G., Prykhod'ko A.O.
- Sapelkin V.,Yakovenko
O.,Golub A., Bdzhola V., Yarmoluk S. Search for protein kinase CK2
inhibitors among 4 aminoquinazoline derivatives. Ukrainica Bioorganica
Acta. – 2004. – 1, ¹ 1-2, 74-79.
- Golub A.G.,
Yakovenko O.Ya., Bdzhola V. G., Yarmoluk S.M. Study of Casein kinase
II inhibitory activity of 4-aminoquinoline and 4-aminoquinazoline
derivatives by combined docking-molecular dynamics approach. Cell.
Mol. Biol. Lett. – Vol. 8, N 2A. – 2003. – P. 584.
- Golub A.G.,
Yakovenko O.Ya., Bdzhola V. G., Yarmoluk S.M. Topbuilder – molecular
topology building and chemical database processing software. Cell.
Mol. Biol. Lett. – Vol. 8, N 2A. – 2003. – P. 610.
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